2
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T2435 | EPZ011989 | Histone Methyltransferase | |
EPZ011989 is a effective, specific orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 Y646 and EZH2 wt; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase. | |||
T2435L | EPZ011989 HCl(1598383-40-4 Free base) | EPZ-011989 TFA,EPZ011989 TFA salt,EPZ 011989 TFA,EPZ011989 TFA | |
EPZ011989 is a highly potent and selective oral EZH2 inhibitor with Ki value <3 nM. |